bitolterol

Term ID

CHEBI:3133

Synonyms

4-(2-(tert-butylamino)-1-hydroxyethyl)-o-phenylene di-p-toluate
4-[2-(tert-butylamino)-1-hydroxyethyl]-o-phenylene di-p-toluate
4-[2-(tert-butylamino)-1-hydroxyethyl]benzene-1,2-diyl bis(4-methylbenzoate)
bis(4-methylbenzoic acid) 4-[2-(tert-butylamino)-1-hydroxyethyl]-1,2-phenylene ester
bitolterol
bitolterolum

Definition

The di-4-toluate ester of (+-)-N-tert-butylnoradrenaline (colterol). A pro-drug for colterol, a beta2-adrenergic receptor agonist, bitolterol is used as its methanesulfonate salt for relief of bronchospasm in conditions such as asthma, chronic bronchitis and emphysema.

References

Beilstein:2229527
CAS:30392-40-6
DrugBank:DB00901
Drug_Central:384
KEGG:C06853
KEGG:D07534
PMID:3278878
PMID:473792
Patent:DE2015573
Patent:US4138581
Reaxys:2229527
Wikipedia:Bitolterol

Ontology

ChEBI ( EBI )

Resources

CTD

Relationships

is a type of: carboxylic ester diester ethanolamines secondary alcohol secondary amino compound

carboxylic ester diester ethanolamines secondary alcohol secondary amino compound Show first 5 Terms
has subtype: (R)-bitolterol (S)-bitolterol

(R)-bitolterol (S)-bitolterol Show first 5 Terms
has_role: anti-asthmatic drug beta-adrenergic agonist bronchodilator agent prodrug

anti-asthmatic drug beta-adrenergic agonist bronchodilator agent prodrug Show first 5 Terms
inverse has_part: bitolterol mesylate

bitolterol mesylate Show first 5 Terms

Phenotype

Phenotype resulting from bitolterol

Phenotype where environments contain bitolterol

Phenotype modified by environments containing bitolterol

Human Disease / Model Data

Citations