Search Ontology:
ChEBI

L-803087

Term ID
CHEBI:177197
Synonyms
  • L 803087
  • L-803,087
  • L803087
  • methyl (2S)-5-carbamimidamido-2-[4-(5,7-difluoro-2-phenyl-1H-indol-3-yl)butanamido]pentanoate
  • methyl N(2)-[4-(5,7-difluoro-2-phenyl-1H-indol-3-yl)butanoyl]-L-argininate
  • N(2)-[4-(5,7-difluoro-2-phenyl-1H-indol-3-yl)-1-oxobutyl]-L-arginine methyl ester
Definition
A fluoroindole that is 1H-indole substituted by phenyl, 4-{[(2S)-5-carbamimidamido-1-methoxy-1-oxopentan-2-yl]amino}-4-oxobutyl, fluoro and fluoro groups at positions 2, 3, 5 and 7, respectively. It is a selective nonpeptidic agonist of the somatostatin subtype-4 (SST4) receptor with Ki of 0.7 nM.
References
  • cas:217480-26-7
  • chemspider:4470867
  • lincs.smallmolecule:LSM-1482
  • pubmed:10433861
  • pubmed:11087999
  • pubmed:12372020
  • pubmed:14667213
  • pubmed:15380378
  • pubmed:15733093
  • pubmed:16081634
  • pubmed:18390640
  • pubmed:18521573
  • pubmed:18766330
  • pubmed:19623609
  • pubmed:19811607
  • pubmed:20573967
  • pubmed:20826222
  • pubmed:21854790
  • pubmed:26631476
  • pubmed:30675231
  • pubmed:9784130
Ontology
ChEBI  ( EBI )
Relationships
Phenotype
Phenotype resulting from L-803087
Phenotype where environments contain L-803087
Phenotype modified by environments containing L-803087
Phenotype affecting L-803087
Human Disease Model