Search Ontology:
ChEBI
kenpaullone
- Term ID
- CHEBI:92658
- Synonyms
-
- 9-bromo-7,12-dihydroindolo[3,2-d][1]benzazepin-6(5H)-one
- 9-bromopaullone
- Definition
- An indolobenzazepine that is paullone in which the hydrogen at position 9 is replaced by a bromo substituent. It is an ATP-competitive inhibitor of cyclin-dependent kinases (CDKs) and glycogen synthase kinase 3beta (GSK3beta).
- References
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- CAS:142273-20-9
- Chemspider:3688
- LINCS:LSM-2824
- PMCID:PMC6216549
- PMCID:PMC8551327
- PMID:10425100
- PMID:16122578
- PMID:16499355
- PMID:24134630
- PMID:24978614
- PMID:25616642
- PMID:27008992
- PMID:28955831
- PMID:29128602
- PMID:29514916
- PMID:29577900
- PMID:30038266
- PMID:31296906
- PMID:31911436
- PMID:33410342
- Reaxys:5346108
- Ontology
- ChEBI ( EBI )
- is a type of
-
- has_functional_parent
-
- has_role
-
Phenotype
Phenotype resulting from kenpaullone
Phenotype where environments contain kenpaullone
Phenotype modified by environments containing kenpaullone
Human Disease Model