Search Ontology:
ChEBI

PQIP

Term ID
CHEBI:90536
Synonyms
  • 3-[cis-3-(4-methylpiperazin-1-yl)cyclobutyl]-1-(2-phenylquinolin-7-yl)imidazo[1,5-a]pyrazin-8-amine
Definition
A member of the class of imidazopyrazines that is imidazo[1,5-a]pyrazin-8-amine carrying additional 2-phenylquinolin-7-yl and 3-(4-methylpiperazin-1-yl)cyclobutyl groups at positions 1 and 3 respectively. It is an inhibitor of insulin growth factor 1 receptor (IGF-1 receptor, IGFR1R) tyrosine kinase.
References
  • pdb-ccd:D94
  • pubmed:17671083
  • pubmed:18566589
  • pubmed:20943761
  • pubmed:21850397
  • pubmed:22101930
  • pubmed:23239200
  • reaxys:12423292
  • reaxys:12923638
Ontology
ChEBI  ( EBI )
Relationships
Phenotype
Phenotype resulting from PQIP
Phenotype where environments contain PQIP
Phenotype modified by environments containing PQIP
Phenotype affecting PQIP
Human Disease Model