Search Ontology:
ChEBI

selumetinib

Term ID
CHEBI:90227
Synonyms
  • 5-[(4-bromo-2-chlorophenyl)amino]-4-fluoro-N-(2-hydroxyethoxy)-1-methyl-1H-benzimidazole-6-carboxamide
  • ARRY 142886
  • ARRY-142886
  • ARRY142886
  • AZD 6244
  • AZD-6244
  • AZD6244
  • selumetinib
  • selumetinibum
Definition
A member of the class of benzimidazoles that is 1-methyl-1H-benzimidazole which is substituted at positions 4, 5, and 6 by fluorine, (4-bromo-2-chlorophenyl)amino, and N-(2-hydroxyethoxy)aminocarbonyl groups, respectively. It is a MEK1 and MEK2 inhibitor.
References
  • cas:606143-52-6
  • kegg.drug:D09666
  • lincs.smallmolecule:LSM-1056
  • pdb-ccd:3EW
  • pubmed:20407895
  • pubmed:20978926
  • pubmed:21594619
  • pubmed:22241789
  • pubmed:22343622
  • pubmed:22394161
  • pubmed:22565394
  • pubmed:22972589
  • pubmed:23372439
  • pubmed:23444215
  • pubmed:23942066
  • pubmed:25322874
  • pubmed:25342139
  • pubmed:25379021
  • pubmed:25385055
  • pubmed:25498501
  • pubmed:25637165
  • pubmed:25887099
  • pubmed:26059332
  • pubmed:26384399
  • pubmed:26446942
  • reaxys:11099648
  • wikipedia.en:Selumetinib
Ontology
ChEBI  ( EBI )
Relationships
Phenotype
Phenotype resulting from selumetinib
Phenotype where environments contain selumetinib
Phenotype modified by environments containing selumetinib
Phenotype affecting selumetinib
Human Disease Model