Search Ontology:
ChEBI

varenicline

Term ID
CHEBI:84500
Synonyms
  • 7,8,9,10-Tetrahydro-6,10-methano-6H-pyrazino(2,3-h)(3)benzazepine
  • 7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g]quinoxaline
  • vareniclina
  • varenicline
  • vareniclinum
Definition
An organic heterotetracyclic compound that acts as a partial agonist for nicotinic cholinergic receptors and is used (in the form of its tartate salt) as an aid to giving up smoking.
References
  • cas:249296-44-4
  • drugbank:DB01273
  • drugcentral:2808
  • hmdb:HMDB0015398
  • kegg.drug:D08669
  • lincs.smallmolecule:LSM-5358
  • pdb-ccd:QMR
  • pubmed:24406270
  • pubmed:24652107
  • pubmed:24763764
  • pubmed:24856597
  • pubmed:24906297
  • pubmed:24949564
  • pubmed:25062287
  • pubmed:25145377
  • pubmed:25331778
  • pubmed:25352081
  • pubmed:25410148
  • pubmed:25449275
  • pubmed:25462656
  • pubmed:25475645
  • pubmed:25485645
  • pubmed:25497715
  • pubmed:25572451
  • pubmed:25588294
  • pubmed:25616031
  • reaxys:10668886
  • wikipedia.en:Varenicline
Ontology
ChEBI  ( EBI )
Relationships
Phenotype
Phenotype resulting from varenicline
Phenotype where environments contain varenicline
Phenotype modified by environments containing varenicline
Phenotype affecting varenicline
Human Disease Model