Search Ontology:
ChEBI

paliperidone palmitate

Term ID
CHEBI:83807
Synonyms
  • (+-)-paliperidone palmitate
  • (RS)-paliperidone palmitate
  • INVEGA SUSTENNA
  • paliperidone hexadecanoate
  • rac-3-{2-[4-(6-fluoro-1,2-benzoxazol-3-yl)piperidin-1-yl]ethyl}-2-methyl-4-oxo-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidin-9-yl hexadecanoate
  • rac-paliperidone palmitate
  • racemic paliperidone palmitate
  • RO 92670
  • RO92670
  • Xeplion
Definition
A racemate comprising equimolar amounts of (R)- and (S)-paliperidone palmitate. A long-acting injectable formulation of paliperidone (the major active metabolite of risperidone) that is used for treatment of schizophrenia.
References
  • cas:199739-10-1
  • kegg.drug:D05340
  • pubmed:22571444
  • pubmed:23237346
  • pubmed:23446197
  • pubmed:24113628
  • pubmed:24117209
  • pubmed:24419004
  • pubmed:24429948
  • pubmed:24559194
  • pubmed:24590546
  • pubmed:24676998
  • pubmed:24754314
  • pubmed:24758296
  • pubmed:24764772
  • pubmed:24845884
  • pubmed:24846035
  • pubmed:24853962
  • pubmed:24882037
  • pubmed:25251693
  • pubmed:25375367
  • reaxys:15026585
  • wikipedia.en:Paliperidone
Ontology
ChEBI  ( EBI )
Relationships
Phenotype
Phenotype resulting from paliperidone palmitate
Phenotype where environments contain paliperidone palmitate
Phenotype modified by environments containing paliperidone palmitate
Phenotype affecting paliperidone palmitate
Human Disease Model