Search Ontology:
ChEBI

riociguat

Term ID
CHEBI:76018
Synonyms
  • Adempas
  • BAY 63-2521
  • Methyl N-(4,6-diamino-2-{1-((2-fluorophenyl)methyl)-1H-pyrazolo(3,4-b)pyridin-3-yl}pyrimidin-5-yl)-N-methylcarbamate
  • methyl {4,6-diamino-2-[1-(2-fluorobenzyl)-1H-pyrazolo[3,4-b]pyridin-3-yl]pyrimidin-5-yl}methylcarbamate
  • riociguat
  • riociguatum
Definition
A carbamate ester that is the methyl ester of {4,6-diamino-2-[1-(2-fluorobenzyl)-1H-pyrazolo[3,4-b]pyridin-3-yl]pyrimidin-5-yl}methylcarbamic acid. It is used for treatment of chronic thromboembolic pulmonary hypertension and pulmonary arterial hypertension
References
  • cas:625115-55-1
  • drugcentral:4807
  • kegg.drug:D09572
  • patent:US2009286781
  • patent:WO2007009607
  • patent:WO2011147810
  • pmc:PMC3363218
  • pubmed:19129292
  • pubmed:20424448
  • pubmed:20801938
  • pubmed:20956169
  • pubmed:21391889
  • pubmed:21789188
  • pubmed:22719060
  • pubmed:22900035
  • pubmed:22912874
  • pubmed:22936711
  • pubmed:23204120
  • pubmed:23397304
  • pubmed:23775260
  • pubmed:23883377
  • pubmed:23883378
  • pubmed:23883383
  • pubmed:23939482
  • pubmed:23963798
  • pubmed:23978639
  • pubmed:23997048
  • pubmed:23997053
  • pubmed:24015306
  • pubmed:24092345
  • reaxys:12581953
  • wikipedia.en:Riociguat
Ontology
ChEBI  ( EBI )
Relationships
Phenotype
Phenotype resulting from riociguat
Phenotype where environments contain riociguat
Phenotype modified by environments containing riociguat
Phenotype affecting riociguat
Human Disease Model