Search Ontology:
ChEBI

lomitapide

Term ID
CHEBI:72297
Synonyms
  • AEGR 733
  • AEGR 773
  • AEGR-773
  • AEGR733
  • AEGR773
  • BMS 201038
  • BMS201038
  • Lojuxta
  • lomitapida
  • lomitapide
  • lomitapidum
  • N-(2,2,2-trifluoroethyl)-9-{4-[4-({[4'-(trifluoromethyl)biphenyl-2-yl]carbonyl}amino)piperidin-1-yl]butyl}-9H-fluorene-9-carboxamide
Definition
A member of the class of benzamides obtained by formal condensation of the carboxy group of 4'-(trifluoromethyl)biphenyl-2-carboxylic acid with the primary amino group of 9-[4-(4-aminopiperidin-1-yl)butyl]-N-(2,2,2-trifluoroethyl)-9H-fluorene-9-carboxamide. Used (as its mesylate salt) as a complement to a low-fat diet and other lipid-lowering treatments in patients with homozygous familial hypercholesterolemia.
References
  • cas:182431-12-5
  • drugbank:DB08827
  • drugcentral:4721
  • kegg.drug:D09637
  • patent:US2003162788
  • patent:US2008161279
  • patent:US2010273829
  • patent:US2011288064
  • patent:US2011288110
  • patent:US2012035204
  • patent:US2012071458
  • pubmed:17215532
  • pubmed:20127562
  • pubmed:21846156
  • pubmed:22963620
  • pubmed:23122767
  • pubmed:23122768
  • pubmed:23147576
  • pubmed:24366202
  • pubmed:25257075
  • pubmed:25702706
  • pubmed:26120010
  • pubmed:26686567
  • pubmed:27055957
  • pubmed:27232459
  • pubmed:27785928
  • pubmed:28154305
  • pubmed:28239069
  • pubmed:28255870
  • pubmed:28432645
  • pubmed:28598687
  • pubmed:28716835
  • reaxys:13754976
  • wikipedia.en:Lomitapide
Ontology
ChEBI  ( EBI )
Relationships
Phenotype
Phenotype resulting from lomitapide
Phenotype where environments contain lomitapide
Phenotype modified by environments containing lomitapide
Phenotype affecting lomitapide
Human Disease Model