Search Ontology:
ChEBI

tofacitinib citrate

Term ID
CHEBI:71197
Synonyms
  • 3-{(3R,4R)-4-methyl-3-[methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrile 2-hydroxypropane-1,2,3-tricarboxylate
  • CP-690,550-10
  • Tasocitinib citrate
  • Xeljanz
Definition
A citrate salt obtained by combining equimolar amounts of tofacitinib and citric acid. Used to treat moderately to severely active Rheumatoid Arthritis.
References
  • cas:540737-29-9
  • kegg.drug:D09783
  • patent:US2003130292
  • patent:WO2005063251
  • patent:WO2005105146
  • pubmed:21105711
  • reaxys:11610699
Ontology
ChEBI  ( EBI )
Relationships
Phenotype
Phenotype resulting from tofacitinib citrate
Phenotype where environments contain tofacitinib citrate
Phenotype modified by environments containing tofacitinib citrate
Phenotype affecting tofacitinib citrate
Human Disease Model