Search Ontology:
ChEBI

lurasidone

Term ID
CHEBI:70735
Synonyms
  • (3aR,4S,7R,7aS)-2-{[(1R,2R)-2-{[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]methyl}cyclohexyl]methyl}hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione
  • lurasidona
  • lurasidone
  • lurasidonum
Definition
An N-arylpiperazine that is (3aR,4S,7R,7aS)-2-{[(1R,2R)-2-(piperazin-1-ylmethyl)cyclohexyl]methyl}hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione in which position N4 of the piperazine ring is substituted by a 1,2-benzothiazol-3-yl group. Lurasidone is used (generally as the hydrochloride salt) as an atypical antipsychotic for the treatment of schizophrenia.
References
  • cas:367514-87-2
  • drugcentral:4168
  • patent:EP1637530
  • patent:EP1652848
  • patent:US2011263847
  • patent:US2011263848
  • patent:US2012115879
  • pubmed:19780705
  • pubmed:21349227
  • pubmed:21474903
  • pubmed:21838595
  • pubmed:22072817
  • pubmed:22217440
  • pubmed:22227609
  • pubmed:22332980
  • pubmed:22364325
  • pubmed:22395527
  • pubmed:22415605
  • pubmed:22545643
  • pubmed:22559286
  • pubmed:22570547
  • pubmed:22675261
  • pubmed:22739469
  • pubmed:22776634
  • pubmed:22828971
  • pubmed:22849428
  • pubmed:22868411
  • pubmed:22900950
  • pubmed:22903391
  • pubmed:22929996
  • pubmed:22967786
  • pubmed:23001538
  • reaxys:11182976
  • wikipedia.en:Lurasidone
Ontology
ChEBI  ( EBI )
Relationships
Phenotype
Phenotype resulting from lurasidone
Phenotype where environments contain lurasidone
Phenotype modified by environments containing lurasidone
Phenotype affecting lurasidone
Human Disease Model