Search Ontology:
ChEBI

(S)-(-)-sulpiride

Term ID
CHEBI:64119
Synonyms
  • (-)-N-(((S)-1-Ethyl-2-pyrrolidinyl)methyl)-5-sulfamoyl-o-anisamide
  • (-)-sulpiride
  • (S)-(-)-5-aminosulfonyl-N-[(1-ethyl-2-pyrrolidinyl)methyl]-2-methoxybenzamide
  • (S)-(-)-N-((1-Ethyl-2-pyrrolidinyl)methyl)-5-sulfamoyl-o-anisamide
  • (S)-sulpiride
  • levosulpirida
  • levosulpiride
  • levosulpiridum
  • N-{[(2S)-1-ethylpyrrolidin-2-yl]methyl}-2-methoxy-5-sulfamoylbenzamide
  • S-(-)-N-(1-Ethyl-2-pyrrolidinomethyl)-2-methoxy-5-sulfamoylebenzamide
Definition
An optically active form of sulpiride having (S)-configuration. The active enantiomer of the racemic drug sulpiride. Selective D2-like dopamine antagonist (Ki values are ~ 0.015. ~ 0.013, 1, ~ 45 and ~ 77 μM at D2, D3, D4, D1 and D5 receptors respectively).
References
  • cas:23672-07-3
  • drugbank:DB00391
  • drugcentral:1577
  • kegg.drug:D07312
  • lincs.smallmolecule:LSM-5624
  • patent:KR20110090142
  • patent:US2011052700
  • pubmed:18186115
  • pubmed:19165957
  • pubmed:19452563
  • pubmed:19488984
  • pubmed:19795476
  • pubmed:20438811
  • pubmed:20656570
  • pubmed:20850200
  • pubmed:21223496
  • pubmed:21615988
  • reaxys:3563418
  • wikipedia.en:Levosulpiride
Ontology
ChEBI  ( EBI )
Resources
CTD
Relationships
Phenotype
Phenotype resulting from (S)-(-)-sulpiride
Phenotype where environments contain (S)-(-)-sulpiride
Phenotype modified by environments containing (S)-(-)-sulpiride
Phenotype affecting (S)-(-)-sulpiride
Human Disease Model