Search Ontology:
ChEBI

labetalol

Term ID
CHEBI:6343
Synonyms
  • 2-hydroxy-5-{1-hydroxy-2-[(1-methyl-3-phenylpropyl)amino]ethyl}benzamide
  • 3-Carboxamido-4-hydroxy-alpha-((1-methyl-3-phenylpropylamino)methyl)benzyl alcohol
  • 5-(1-Hydroxy-2-(1-methyl-3-phenylpropylamino)ethyl)salicylamide
  • kabetalol
  • labetalol
  • labetalolum
Definition
A diastereoisomeric mixture of approximately equal amounts of all four possible stereoisomers ((R,S)-labetolol, (S,R)-labetolol, (S,S)-labetalol and (R,R)-labetalol). It is an adrenergic antagonist used to treat high blood pressure.
References
  • cas:36894-69-6
  • drugbank:DB00598
  • drugcentral:1531
  • hmdb:HMDB0014736
  • kegg.compound:C07063
  • kegg.drug:D08106
  • lincs.smallmolecule:LSM-1282
  • patent:DE2032642
  • patent:US4012444
  • pubmed:1447344
  • pubmed:16795017
  • pubmed:21908132
  • pubmed:22300487
  • pubmed:22528277
  • pubmed:23055089
  • pubmed:28166217
  • pubmed:31643185
  • pubmed:32709242
  • pubmed:33210850
  • pubmed:33424327
  • pubmed:33638710
  • pubmed:33893609
  • pubmed:34217067
  • pubmed:35075411
  • pubmed:7295463
  • reaxys:2948416
  • wikipedia.en:Labetalol
Ontology
ChEBI  ( EBI )
Resources
CTD
Relationships
Phenotype
Phenotype resulting from labetalol
Phenotype where environments contain labetalol
Phenotype modified by environments containing labetalol
Phenotype affecting labetalol
Human Disease Model