Search Ontology:
ChEBI

E3040

Term ID
CHEBI:4732
Synonyms
  • 5,7-dimethyl-2-(methylamino)-4-(pyridin-3-ylmethyl)-1,3-benzothiazol-6-ol
  • 6-hydroxy-5,7-dimethyl-2-methylamino-4-(3-pyridylmethyl) benzothiazole
  • E-3040
  • E3040
Definition
A member of the class of benzothiazoles that is 1,3-benzothiazole substituted by a methylnitrilo group, (pyridin-3-yl)methyl group, methyl group, hydroxy group and methyl group at position 2,4,5,6 and 7, respectively. It is a dual inhibitor of 5-lipoxygenase and thromboxane A2 synthetase and exhibits anti-inflammatory properties. The drug was being developed by Eisai (Tokyo, Japan) for the treatment of bowel disease.
References
  • cas:145096-30-6
  • kegg.compound:C11593
  • pubmed:10206322
  • pubmed:10594872
  • pubmed:11011031
  • pubmed:11430933
  • pubmed:11557269
  • pubmed:12023941
  • pubmed:15319327
  • pubmed:15598971
  • pubmed:7562509
  • pubmed:8536337
  • pubmed:8592681
  • pubmed:9023311
  • pubmed:9262353
Ontology
ChEBI  ( EBI )
Resources
CTD
Relationships
Phenotype
Phenotype resulting from E3040
Phenotype where environments contain E3040
Phenotype modified by environments containing E3040
Phenotype affecting E3040
Human Disease Model