Search Ontology:
ChEBI

imatinib methanesulfonate

Term ID
CHEBI:31690
Synonyms
  • 4-[(4-methylpiperazin-1-yl)methyl]-N-{4-methyl-3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl}benzamide methanesulfonate
  • Gleevec
  • Glivec
  • imatinib mesilate
  • imatinib mesylate
  • imatinib methansulfonate
  • imatinib monomesylate
Definition
A methanesulfonate (mesylate) salt that is the monomesylate salt of imatinib. Used for treatment of chronic myelogenous leukemia and gastrointestinal stromal tumours.
References
  • cas:220127-57-1
  • drugbank:DB00619
  • hmdb:HMDB0014757
  • kegg.drug:D01441
  • patent:RU2365587
  • patent:WO2004106326
  • patent:WO2011161689
  • patent:WO9903854
  • pubmed:12047970
  • pubmed:12616857
  • pubmed:12669406
  • pubmed:12975485
  • pubmed:14760091
  • pubmed:15059881
  • pubmed:15161340
  • pubmed:15206509
  • pubmed:15250677
  • pubmed:15601563
  • pubmed:15727903
  • pubmed:16570351
  • pubmed:16805961
  • pubmed:16835496
  • pubmed:17212133
  • pubmed:18422477
  • pubmed:19073506
  • pubmed:19258052
  • pubmed:19508953
  • pubmed:19542718
  • pubmed:19568828
  • pubmed:21084823
  • pubmed:21333826
  • pubmed:23462796
  • reaxys:10229624
Ontology
ChEBI  ( EBI )
Relationships
Phenotype
Phenotype resulting from imatinib methanesulfonate
Phenotype where environments contain imatinib methanesulfonate
Phenotype modified by environments containing imatinib methanesulfonate
Phenotype affecting imatinib methanesulfonate
Human Disease Model