Search Ontology:
ChEBI

tebanicline

Term ID
CHEBI:234304
Synonyms
  • (R)-5-(2-azetidinylmethoxy)-2-chloropyridine
  • (R)-5-(azetidin-2-ylmethoxy)-2-chloropyridine
  • 5-((2R)-azetidinylmethoxy)-2-chloropyridine
  • 5-[((2R)-azetidin-2-yl)methoxy]-2-chloropyridine
  • 5-[(2R)-2-azetidinylmethoxy]-2-chloropyridine
  • 5-[(2R)-azetidin-2-ylmethoxy]-2-chloropyridine
  • ABT 594
  • ABT-594
  • ABT594
  • ebanicline
  • tebaniclina
  • tebanicline
  • tebaniclinum
Definition
A monochloropyridine that is 2-chloropyridine substituted by a (2R)-azetidin-2-ylmethoxy group at position 5. It is a potent nicotinic acetylcholine receptor agonist with analgesic and antinociceptive properties.
References
  • cas:198283-73-7
  • patent:WO9953922
  • pubmed:10716232
  • pubmed:10779668
  • pubmed:10781917
  • pubmed:14682326
  • pubmed:15072432
  • pubmed:15542623
  • pubmed:15713428
  • pubmed:16289887
  • pubmed:16412637
  • pubmed:17706609
  • pubmed:18088559
  • pubmed:19232492
  • pubmed:19632048
  • pubmed:20064548
  • pubmed:20562022
  • pubmed:21620806
  • pubmed:22145610
  • pubmed:22328206
  • pubmed:23925734
  • pubmed:27939354
  • pubmed:29332255
  • pubmed:30222192
  • pubmed:32294065
  • pubmed:40175361
  • pubmed:9417028
  • pubmed:9484491
  • pubmed:9580626
  • pubmed:9580627
  • pubmed:9617748
  • pubmed:9651224
  • pubmed:9729357
  • pubmed:9789812
  • wikipedia.en:Tebanicline
Ontology
ChEBI  ( EBI )
Relationships
Phenotype
Phenotype resulting from tebanicline
Phenotype where environments contain tebanicline
Phenotype modified by environments containing tebanicline
Phenotype affecting tebanicline
Human Disease Model