Search Ontology:
ChEBI

KU-60019

Term ID
CHEBI:228206
Synonyms
  • 2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-{5-[6-(morpholin-4-yl)-4-oxo-4H-pyran-2-yl]-9H-thioxanthen-2-yl}acetamide
  • KU 60019
  • KU60019
Definition
A secondary carboxamide resulting from the formal condensation of the carboxy group of [(2R,6S)-2,6-dimethylmorpholin-4-yl]acetic acid with the amino group of 2-(7-amino-9H-thioxanthen-4-yl)-6-(morpholin-4-yl)-4H-pyran-4-one. It is an ATM kinase inhibitor (IC50 = 6.3 nM).
References
  • cas:925701-46-8
  • cas:925701-49-1
  • lincs.smallmolecule:LSM-1156
  • pubmed:19808981
  • pubmed:23620409
  • pubmed:24443327
  • pubmed:25091220
  • pubmed:25289090
  • pubmed:26620371
  • pubmed:28693235
  • pubmed:29522753
  • pubmed:31299316
  • pubmed:31597711
  • pubmed:31626963
  • pubmed:33971260
  • pubmed:34433825
  • pubmed:35477555
  • pubmed:35734412
  • pubmed:35783188
  • pubmed:35795059
  • pubmed:35835838
  • pubmed:36228747
  • pubmed:36314821
  • pubmed:36510329
  • pubmed:36650267
  • pubmed:36941082
  • pubmed:37620619
Ontology
ChEBI  ( EBI )
Relationships
Phenotype
Phenotype resulting from KU-60019
Phenotype where environments contain KU-60019
Phenotype modified by environments containing KU-60019
Phenotype affecting KU-60019
Human Disease Model