Search Ontology:
ChEBI

varespladib methyl

Term ID
CHEBI:192805
Synonyms
  • A-002
  • LY 333013
  • LY-333013
  • LY333013
  • methyl ({3-[amino(oxo)acetyl]-1-benzyl-2-ethyl-1H-indol-4-yl}oxy)acetate
  • methyl varespladib
  • methyl-varespladib
  • S 3013
  • S-3013
  • S3013
  • varespladib methyl ester
  • varespladib-methyl
Definition
A methyl ester resulting from the formal condensation of the carboxy group of varespladib with methanol. It is a potential therapy for the treatment of snakebite envenomings in which toxicity depends on the action of PLA2s.
References
  • cas:172733-08-3
  • chemspider:8062590
  • drugbank:DB05737
  • hmdb:HMDB0259767
  • kegg.drug:D08221
  • pubmed:15742431
  • pubmed:19697278
  • pubmed:20809869
  • pubmed:20863951
  • pubmed:21174506
  • pubmed:21446779
  • pubmed:21989792
  • pubmed:27571102
  • pubmed:30241297
  • pubmed:30453607
  • pubmed:31146670
  • pubmed:31226842
  • pubmed:32093386
  • pubmed:32560391
  • pubmed:32889027
  • pubmed:34143707
Ontology
ChEBI  ( EBI )
Relationships
Phenotype
Phenotype resulting from varespladib methyl
Phenotype where environments contain varespladib methyl
Phenotype modified by environments containing varespladib methyl
Phenotype affecting varespladib methyl
Human Disease Model