Search Ontology:
ChEBI

arachidonyl-2'-chloroethylamide

Term ID
CHEBI:191854
Synonyms
  • (5Z,8Z,11Z,14Z)-N-(2-chloroethyl)-5,8,11,14-eicosatetraenamide
  • (5Z,8Z,11Z,14Z)-N-(2-chloroethyl)icosa-5,8,11,14-tetraenamide
  • ACEA
  • arachidonyl-2-chloroethylamide
  • N-(2-chloroethyl)-5Z,8Z,11Z,14Z-eicosatetraenamide
Definition
A fatty amide obtained by the formal condensation of arachidonic acid with 2-chloroethanamine. It is a potent agonist of the CB1 receptor (Ki = 1.4 nM) and also has a low affinity for the CB2 receptor (Ki = 3100 nM).
References
  • cas:220556-69-4
  • chemspider:4470547
  • hmdb:HMDB0247891
  • pubmed:10336536
  • pubmed:12095655
  • pubmed:15006899
  • pubmed:15277316
  • pubmed:15493300
  • pubmed:16649551
  • pubmed:16930590
  • pubmed:18362599
  • pubmed:19751793
  • pubmed:25881484
  • pubmed:25904357
  • pubmed:26820679
  • pubmed:27663280
  • pubmed:28441341
  • pubmed:28859122
  • pubmed:30552944
  • pubmed:30607903
  • pubmed:32413434
  • pubmed:33083022
  • pubmed:33220269
  • pubmed:34090883
  • pubmed:35189809
  • wikipedia.en:Arachidonyl-2'-chloroethylamide
Ontology
ChEBI  ( EBI )
Relationships
Phenotype
Phenotype resulting from arachidonyl-2'-chloroethylamide
Phenotype where environments contain arachidonyl-2'-chloroethylamide
Phenotype modified by environments containing arachidonyl-2'-chloroethylamide
Phenotype affecting arachidonyl-2'-chloroethylamide
Human Disease Model