pelabresib

Term ID

CHEBI:189653

Synonyms

2-((4S)-6-(4-chlorophenyl)-1-methyl-4H-isoxazolo[5,4-d][2]benzazepin-4-yl)acetamide
2-[(4S)-6-(4-chlorophenyl)-1-methyl-4H-[1,2]oxazolo[5,4-d][2]benzazepin-4-yl]acetamide
CPI 0610
CPI-0610
CPI-0610 anhydrous
CPI-232
CPI0610
pelabresib
pelabresibum

Definition

An organic heterotricyclic compound that is 4H-[1,2]oxazolo[5,4-d][2]benzazepine substituted by methyl, 2-amino-2-oxoethyl, and 4-chlorophenyl groups at positions 1, 4S and 6, respectively. It is a small molecule inhibitor of bromodomain and extra-terminal (BET) proteins and exhibits antineoplastic activity.

References

Ontology

ChEBI ( EBI )

Relationships

is a type of: monochlorobenzenes organic heterotricyclic compound primary carboxamide

monochlorobenzenes organic heterotricyclic compound primary carboxamide Show first 5 Terms
has_role: antineoplastic agent bromodomain-containing protein 4 inhibitor

antineoplastic agent bromodomain-containing protein 4 inhibitor Show first 5 Terms

Phenotype

Phenotype resulting from pelabresib

Phenotype where environments contain pelabresib

Phenotype modified by environments containing pelabresib

Human Disease / Model Data