Search Ontology:
ChEBI

NSC 23766

Term ID
CHEBI:144984
Synonyms
  • N(6)-(2-{[5-(diethylamino)pentan-2-yl]amino}-6-methylpyrimidin-4-yl)-2-methylquinoline-4,6-diamine
  • N6-[2-[5-(diethylamino)pentan-2-ylamino]-6-methyl-4-pyrimidinyl]-2-methylquinoline-4,6-diamine
  • NSC-23766
  • NSC23766
Definition
An aminopyrimidine that is 6-methylpyrimidine-2,4-diamine in which the amino groups at positions 2 and 4 are substituted by 5-(diethylamino)pentan-2-yl and 4-amino-2-methylquinolin-6-yl groups respectively. An inhibitor of the signalling G-protein known as RAC1 (Ras-related C3 botulinum toxin substrate 1).
References
  • lincs.smallmolecule:LSM-1818
  • pubmed:15128949
  • pubmed:18183417
  • pubmed:19052208
  • pubmed:19491337
  • pubmed:20515940
  • pubmed:21511011
  • pubmed:23887096
  • pubmed:24257023
  • pubmed:24523909
  • pubmed:24953831
  • pubmed:25154784
  • pubmed:25319697
  • pubmed:25628054
  • pubmed:25631101
  • pubmed:27467102
  • pubmed:29050986
  • pubmed:30871916
Ontology
ChEBI  ( EBI )
Relationships
Phenotype
Phenotype resulting from NSC 23766
Phenotype where environments contain NSC 23766
Phenotype modified by environments containing NSC 23766
Phenotype affecting NSC 23766
Human Disease Model