Search Ontology:
ChEBI

arterolane

Term ID
CHEBI:136054
Synonyms
  • arterolane
  • arterolano
  • arterolanum
  • N-(2-amino-2-methylpropyl)-2-[(1s,4s)-dispiro[cyclohexane-1,3'-[1,2,4]trioxolane-5',2''-tricyclo[3.3.1.1(3,7)]decan]-4-yl]acetamide
  • OZ 277
  • OZ277
  • RBx-11160
  • RBx11160
Definition
An oxaspiro compound that is dispiro[cyclohexane-1,3'-[1,2,4]trioxolane-5',2''-tricyclo[3.3.1.13,7]decane] substituted by a 2-[(2-amino-2-methylpropyl)amino]-2-oxoethyl group at position 4s. Its maleic acid salt is used as an antimalarial drug in combination with piperaquine.
References
  • cas:664338-39-0
  • drugcentral:5090
  • pubmed:15318224
  • pubmed:17087929
  • pubmed:17145800
  • pubmed:17562801
  • pubmed:19646936
  • pubmed:19924861
  • pubmed:20028825
  • pubmed:21814428
  • pubmed:23368889
  • pubmed:23489135
  • pubmed:24242999
  • pubmed:25049252
  • pubmed:25221689
  • pubmed:25530543
  • pubmed:26819968
  • pubmed:27161632
  • pubmed:28052200
  • pubmed:28122617
  • pubmed:28400526
  • pubmed:29263074
  • pubmed:32361471
  • pubmed:32369341
  • wikipedia.en:Arterolane
Ontology
ChEBI  ( EBI )
Relationships
Phenotype
Phenotype resulting from arterolane
Phenotype where environments contain arterolane
Phenotype modified by environments containing arterolane
Phenotype affecting arterolane
Human Disease Model