OBO ID: CHEBI:64111 |
Term Name: | GR 127935 hydrochloride | Search Ontology: | |
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Definition: | A hydrochloride obtained by reaction of GR 127935 with one equivalent of hydrochloric acid. Potent and selective 5-HT1B/1D receptor antagonist (pKi values are 8.5 for both guinea pig 5-HT1D and rat 5-HT1B receptors). Displays > 100-fold selectivity over 5HT1A, 5-HT2A, 5-HT2C receptors and other receptor types. Centrally active following oral administration. | ||
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Ontology: | ChEBI ( EBI ) |
PHENOTYPE
No data available