PUBLICATION

Acetylation of Cavin-1 Promotes Lipolysis in White Adipose Tissue

Authors
Zhou, S.R., Guo, L., Wang, X., Liu, Y., Peng, W.Q., Liu, Y., Wei, X.B., Dou, X., Ding, M., Lei, Q.Y., Qian, S.W., Li, X., Tang, Q.Q.
ID
ZDB-PUB-170601-5
Date
2017
Source
Molecular and cellular biology   37(16): e00058-17 (Journal)
Registered Authors
Wang, Xu
Keywords
WAT, cavin-1, acetylation, HSL, lipolysis
MeSH Terms
  • Cell Membrane/drug effects
  • Cell Membrane/metabolism
  • Protein Binding/drug effects
  • p300-CBP Transcription Factors/metabolism
  • Acetylation/drug effects
  • Lysine/metabolism
  • Animals
  • Mice, Inbred C57BL
  • HEK293 Cells
  • RNA-Binding Proteins/chemistry
  • RNA-Binding Proteins/metabolism*
  • Lipolysis*/drug effects
  • Sirtuin 1/metabolism
  • Humans
  • Lipase/metabolism
  • Mice
  • Male
  • Niacinamide/pharmacology
  • Membrane Proteins/chemistry
  • Membrane Proteins/metabolism*
  • Amino Acid Sequence
  • Adipose Tissue, White/drug effects
  • Adipose Tissue, White/metabolism*
  • 3T3-L1 Cells
  • Zebrafish
PubMed
28559430 Full text @ Mol. Cell. Biol.
Abstract
White adipose tissue (WAT) serves as a reversible energy storage depot in the form of lipids in response to nutritional status. Cavin-1, an essential component in the biogenesis of caveolae, is a positive regulator of lipolysis in adipocytes. However, molecular mechanisms of cavin-1 in the modulation of lipolysis remain poorly understood. Here, we showed that cavin-1 was acetylated at lysines 291, 293, and 298 (3K), which was under nutritional regulation in WAT. We further identified GCN5 as the acetyltransferase and Sirt1 as the deacetylase of cavin-1. Acetylation-mimetic 3Q mutants of cavin-1 augmented fat mobilization in 3T3-L1 adipocytes and zebrafish. Mechanistically, acetylated cavin-1 preferentially interacted with hormone-sensitive lipase and recruited it to the caveolae, thereby promoting lipolysis. Our finding shed light on essential role of cavin-1 in regulating lipolysis via an acetylation-dependent manner in WAT.
Genes / Markers
Figures
Expression
Phenotype
Mutations / Transgenics
Human Disease / Model
Sequence Targeting Reagents
Fish
Antibodies
Orthology
Engineered Foreign Genes
Mapping