PUBLICATION

Mutations in the human SIX3 gene in holoprosencephaly are loss-of-function

Authors
Domené, S., Roessler, E., El-Jaick, K.B., Snir, M., Brown, J.L., Vélez, J.I., Bale, S., Lacbawan, F., Muenke, M., and Feldman, B.
ID
ZDB-PUB-080922-4
Date
2008
Source
Human molecular genetics   17(24): 3919-3928 (Journal)
Registered Authors
Feldman, Benjamin
Keywords
none
MeSH Terms
  • Alleles
  • Amino Acid Motifs/genetics
  • Amino Acid Sequence
  • Amino Acid Substitution/genetics
  • Animals
  • DNA Mutational Analysis
  • Eye Proteins/genetics*
  • Eye Proteins/physiology
  • Holoprosencephaly/etiology
  • Holoprosencephaly/genetics*
  • Holoprosencephaly/metabolism*
  • Homeodomain Proteins/genetics*
  • Homeodomain Proteins/physiology
  • Humans
  • Molecular Sequence Data
  • Nerve Tissue Proteins/genetics*
  • Nerve Tissue Proteins/physiology
  • Point Mutation/genetics*
  • Zebrafish/embryology
  • Zebrafish/genetics
  • Zebrafish/metabolism
PubMed
18791198 Full text @ Hum. Mol. Genet.
Abstract
Holoprosencephaly (HPE) is the most common developmental anomaly of the human forebrain; however, the genetics of this heterogeneous and etiologically complex malformation is incompletely understood. Heterozygous mutations in SIX3, a transcription factor gene expressed in the anterior forebrain and eyes during early vertebrate development, have been frequently detected in human HPE cases. However, only a few mutations have been investigated with limited functional studies that would confirm a role in HPE pathogenesis. Here we report the development of a set of robust and sensitive assays of human SIX3 function in zebrafish, and apply these to the analysis of a total of 46 distinct mutations (19 previously published and 27 novel) located throughout the entire SIX3 gene. We can now confirm that 89% of these putative deleterious mutations are significant loss-of-function alleles. Since disease-associated single point mutations in the Groucho-binding eh1-like motif decreases function in all assays we can also confirm that this interaction is essential for human SIX3 co-repressor activity; we infer, in turn, that this function is important in HPE causation. We also unexpectedly detected truncated versions with partial function, yet missing a SIX3-encoded homeodomain. Our data indicate that SIX3 is a frequent target in the pathogenesis of HPE and demonstrate how this can inform the genetic counseling of families.
Genes / Markers
Figures
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Expression
Phenotype
Mutations / Transgenics
Human Disease / Model
Sequence Targeting Reagents
Fish
Antibodies
Orthology
Engineered Foreign Genes
Mapping