Search Ontology:
ChEBI

regorafenib

Term ID
CHEBI:68647
Synonyms
  • 4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamoyl}amino)-3-fluorophenoxy]-N-methylpyridine-2-carboxamide
  • BAY 73-4506
  • regorafenib
  • regorafenibum
Definition
A pyridinecarboxamide obtained by condensation of 4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamoyl}amino)-3-fluorophenoxy]pyridine-2-carboxylic acid with methylamine. Used for for the treatment of metastatic colorectal cancer in patients who have previously received chemotherapy, anti-EGFR or anti-VEGF therapy.
References
  • cas:755037-03-7
  • drugcentral:4654
  • kegg.drug:D10138
  • lincs.smallmolecule:LSM-1226
  • patent:US2006058358
  • patent:WO2006125540
  • patent:WO2007054216
  • patent:WO2007068380
  • patent:WO2007068382
  • patent:WO2008043446
  • patent:WO2008055629
  • patent:WO2008058644
  • patent:WO2008089388
  • patent:WO2008089389
  • patent:WO2011128261
  • patent:WO2011130728
  • pubmed:21170960
  • pubmed:21419931
  • pubmed:21752724
  • pubmed:22421192
  • pubmed:22568966
  • pubmed:22577890
  • pubmed:22612461
  • pubmed:22614970
  • pubmed:22706543
  • pubmed:22777740
  • pubmed:22785409
  • pubmed:22959186
  • reaxys:14359949
  • wikipedia.en:Regorafenib
Ontology
ChEBI  ( EBI )
Relationships
Phenotype
Phenotype resulting from regorafenib
Phenotype where environments contain regorafenib
Phenotype modified by environments containing regorafenib
Phenotype affecting regorafenib
Human Disease Model