Term Name: GABA modulator
Synonyms: GABA modulators
Definition: A substance that does not act as agonist or antagonist but does affect the gamma-aminobutyric acid receptor-ionophore complex. GABA-A receptors appear to have at least three allosteric sites at which modulators act: a site at which benzodiazepines act by increasing the opening frequency of gamma-aminobutyric acid-activated chloride channels; a site at which barbiturates act to prolong the duration of channel opening; and a site at which some steroids may act.
Ontology: ChEBI [CHEBI:50268]  ( EBI )

Relationships
is a type of: GABA agent membrane transport modulator
inverse has_role: 5alpha-dihydrodeoxycorticosterone alpha-asarone barbiturates benzodiazepine beta-asarone brexanolone clobazam clonazepam clorazepic acid dipotassium clorazepate estazolam isoliquiritigenin nimetazepam nitrazepam nordazepam pinocarveol secobarbital secobarbital sodium valerenic acid verruculogen zuranolone